This post picks up from a few missives ago (Mitigating Heterocyclic Metabolism, Part One) when I was pointing out the fantastic St. Jean and Fotsch Perspective article “Mitigating heterocycle metabolism in drug discovery” [Journal of Medicinal Chemistry 2012, 55(13), 6002-6020]. If you didn’t get a chance to read it, please feel free to examine my […]
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